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Citation: Feng Xiaoming, Jiang Yaozhong, Chen Rong, Ming Liguo. Synthesis of 2-Afoylamino-5-(1-phenyl-2-hydroxyanisethyl)-1,3,4-thiadiazoles[J]. Chinese Journal of Applied Chemistry, ;1994, 44(5): 79-82. shu

Synthesis of 2-Afoylamino-5-(1-phenyl-2-hydroxyanisethyl)-1,3,4-thiadiazoles

1.
1. Chengdu Institute of Organic Chemistry, Chinese Academy of Sciences, Chengdu 610015;
2.
2. Department of Chemistry, Southwest Normal University, Chongqing

Received Date: 31 January 1994
Available Online: 23 March 1994

Thirteen title compounds (2) were obtained by nucleophilic addition of benzyl car-banion of 2-aroylamino-5-benzyl-1,3,4-thiadiazoles (1) with anisaldehyde in EtONa/EtOH solution.The structures of the compounds 2 were confirmed by elemental analysis,IR,¹H NMR,and MS.The compounds were found to have some fungicidal activity.
- thiadiazole,
- nucleophilic addition,
- fungicidal activity
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