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Citation: ZHU Chen-Jiang, SHI Yan, LV Xia, TANG Yan-Hui, CHEN Guo-Rong. Synthesis of Novel Arbutin C-glycoside Derivates and Their Inhibition to Tyrosinase[J]. Chinese Journal of Applied Chemistry, ;2009, 26(3): 253-256. shu

Synthesis of Novel Arbutin C-glycoside Derivates and Their Inhibition to Tyrosinase

1.
Laboratory for Advanced Materials, Institute of Fine Chemicals, East China University of Science and Technology, Shanghai 200237

Corresponding author: CHEN Guo-Rong,
Received Date: 14 February 2008
Available Online: 14 June 2008
Fund Project: 国家自然科学基金(20576034) (20576034)上海市自然科学基金(05ZR14040)资助项目 (05ZR14040)

A series of stable and effective 4-hydroxyphenyl-D-glucopyranoside derivates were synthesized.The 10 new compounds were characterized by ¹H NMR and HRMS.The preliminary test of bioactivity showed that they displayed notable inhibitions to tyrosinase.The inhibitions of compounds 13,14,15,16 and 19 to tyrosinase were equal or better than that of natural arbutin.
- arbutin,
- C-glycoside,
- synthesis,
- inhibitions for tyrosinase
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