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Citation: Li Zaiguo, Huang Runqiu, Yang Zhao, Shao Ruilian. Synthesis and Biological Activity of Diphenyl N-(2-Benzothiazolyl)-α-aminoalkylphosphonate[J]. Chinese Journal of Applied Chemistry, ;1999, 16(2): 94-96. shu

Synthesis and Biological Activity of Diphenyl N-(2-Benzothiazolyl)-α-aminoalkylphosphonate

1.
Institute of Elemento-organic Chemistry, State Key Laboratory of Elemento-organic Chemistry, Nankai University, Tianjin 300071

Received Date: 3 August 1998
Available Online: 7 January 1999
Fund Project: 国家自然科学基金资助课题(29832050) (29832050)

A series of α-(2-benzothiazolyl)-aminoalkyl-phosphonic acid diphenyl esters were synthesized from 2-aminobenzothiazole with aldehyde and triphenyl phosphite.The experiments indicated that the reaction proceeded through the addition of imine with diphenyl phosphite.The bioassy results showed that the compounds have good anti-TMV (tobacco mosaic virus) activities.
- amino(benzo)thiazole,
- α-aminoalkylphosphonic acid diphenyl ester,
- triphenyl hosphite,
- synthesis,
- anti-tobacco mosaic virus activity
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