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Citation: Liu Xin, Huang Runqiu, Li Huiying, Yang Zhao. Synthesis and Bioactivity of O-(4-quinazolinyl) Hydroximic Thioesters (amides)[J]. Chinese Journal of Applied Chemistry, ;1999, 16(2): 27-30. shu

Synthesis and Bioactivity of O-(4-quinazolinyl) Hydroximic Thioesters (amides)

1.
Institute of Elementoorganic Chemistry, State Key Laboratory of Elementoorganic Chemistry, Nankai University, Tianjin 300071

Received Date: 20 July 1998
Available Online: 18 January 1999
Fund Project: 国家自然科学重点基金资助课题(29832050) (29832050)

A series of O-(4-quinazolinyl)hydroximic thioesters(amides) were synthesized by a phase transfer catalysis method. The compounds were found to have good stabilities and antiphy-toviral activities. Some compounds had higher activities against tobacco mosaic virus than 2,4-dioxohexahydro-1,3,5-triazine.
- hydroximic thioester,
- hydroximic thioamide,
- quinazoline,
- synthesis,
- plant virucide
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