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Citation: ZHAO Wei-Guang, CAO Yi-Bing, LI Zheng-Ming, GAO Fa-Wang, WANG Su-Hua, WANG Jian-Guo. Synthesis and Biological Activity of 1-Sulfonyl-3, 5-diamino-1H-Pyrazole Derivatives[J]. Chinese Journal of Applied Chemistry, ;2001, 18(6): 423-427. shu

Synthesis and Biological Activity of 1-Sulfonyl-3, 5-diamino-1H-Pyrazole Derivatives

1.
Institute of Elemento-Organic Chemistry, Nankai University, Tianjin 300071

Received Date: 22 August 2000
Available Online: 9 January 2001
Fund Project: 国家自然科学重点基金资助项目(29832050) (29832050)

1-sulfonyl-3,5-diamino-1H-pyrazole-4-nitriles (3) were synthesized by the reaction of sulfonylation of 3,5-diamino-1H-pyrazole-4-nitriles (2), which were prepared from 2-cyano-3,3-dimethylthio acrylonitrile as starting material with arylamines. All the novel compounds were confirmed by ¹H NMR and elemental analysis, and some by IR and MS. Some of the target compounds show excellent herbicidal activities.
- sulfonylpy razole,
- synthesis,
- herbicide
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