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Citation: MA Ning, LI Zheng-Ming, LI Yong-Hong, HAO Jing-Jun, FAN Chuan-Wen, WANG Ling-Xiu, WANG Su-Hua. Synthesis and Herbicidal Activity of Sulfonylurea Derivatives[J]. Chinese Journal of Applied Chemistry, ;2004, 21(10): 989-992. shu

Synthesis and Herbicidal Activity of Sulfonylurea Derivatives

1.
a State Key Laboratory of Elemento Organic Chemistry, Institute of Elemento Organic Chemistry, Nankai University, Tianjin 300071;
2.
b Department of Chemistry, Tianjin University, Tianjin

Corresponding author: LI Zheng-Ming,
Received Date: 1 December 2003
Available Online: 28 March 2004
Fund Project: 国家"九七三"项目(2003CB114406) (2003CB114406)天津市自然科学重点基金(033803411)资助课题 (033803411)

Alkoxy group and fluorine atom were introduced onto the carbon chain of the substituent of the pyrimidine ring, and 12 novel sulfonylurea compounds with mono substituent in the pyrimidine ring were synthesized. The structures of all compounds were confirmed by ¹H NMR and elemental analysis. Herbicidal activity tests including IC₅₀ in rape root and pot experiments were carried out. The results show that the herbicidal activity decreases as the hydrogen atoms of the alkoxy group at 4-position of the pyrimidine ring are substituted by alkyl, alkoxy groups or fluorine atoms.
- sulfonylurea,
- pyrimidine,
- synthesize,
- herbicide
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