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Citation: WANG Lin, LI Ru-Lin, WANG Hong-Wei, XING Wen-Ru, LIU Wen-Min, YANG Qi-Chao. Synthesis and Biological Activity of N,N'-Naphthalene Acyl Substituted Aromatic Acylamino Thiocarbamides[J]. Chinese Journal of Applied Chemistry, ;2007, 24(10): 1145-1148. shu

Synthesis and Biological Activity of N,N'-Naphthalene Acyl Substituted Aromatic Acylamino Thiocarbamides

1.
a Department of Chemistry, Nanyang Normal College, Nanyang, 473061;
2.
b Department of Biochemistry, Nanyang Institute of Technology, Nanyang

Corresponding author: WANG Lin,
Received Date: 12 November 2006
Available Online: 25 January 2007
Fund Project: 河南省教育厅自然科学研究项目(2003150004) (2003150004)

Eight novel N,N'-naphthalene acyl substituted aromatic acylamino thiocarbamides(Ⅱ₁~Ⅱ₈) were synthesized from aryl acylhydrazine(Ⅰ) and α-naphthalene acyl isothiocyanate, which was obtained by the reaction of potassium thiocyanate with α-naphthalene acyl chloride obtained from 2-naphthylacetic acid and thionyl chloride in anhydrous benzene. The structures of the products were characterized by IR,¹H NMR and elemental analysis. The preliminary biological activity test indicated that the synthesized compounds could promote the growth of paddy root with best effect at 1 mg/L, but had no obvious inhibition activity against B.subtiles and E.coli.
- α-naphthalene acyl,
- substituted aromatic acylamino,
- thiocarbamide,
- synthesis,
- biological activity
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