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Citation: CHEN Chuan-Bing, ZHANG Zheng-Wen, WANG Yan-Gang. Synthesis and Biological Activity of N-(1,3,4-Thiodiazol-2-yl)-N'-aryloxyacetyl Ureas[J]. Chinese Journal of Applied Chemistry, ;2008, 25(7): 862-864. shu

Synthesis and Biological Activity of N-(1,3,4-Thiodiazol-2-yl)-N'-aryloxyacetyl Ureas

1.
a College of Chemistry, Central China Normal University, Wuhan 430079;
2.
b College of traditional Chinese medicine, Guangzhou University of TCM, Guangzhou 510405

Corresponding author: WANG Yan-Gang,
Received Date: 14 July 2007
Available Online: 27 October 2007
Fund Project: 国家自然科学基金资助项目(20072009) (20072009)

Eleven new aryloxyacetyl ureas were synthesized by the reaction of 2-amino-1,3,4-thiodiazole with aryloxyacetyl isocynates in yields of 50.2%~68.7%.Their structures were confirmed by IR,¹H NMR and elemental analysis.The preliminary biological activity tests show that some target compounds have good activities as plant growth regulator.Compounds 2d,2e,2k have a relatively good activity of auxin and the promoting rates of them are 40.1%,35.5% and 28.8% respectively.
- amino-thiodiazole,
- aryloxyacetyl urea,
- synthesis,
- biological activity,
- auxin
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