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Citation: Ying Duan, Yanliang Yang, Xiaoyu Dai, Dongmi Li. Selective arylation/annulation cascade reactions of 2-alkynylanilines with diaryliodonium salts[J]. Chinese Journal of Catalysis, ;2016, 37(11): 1837-1840. doi: 10.1016/S1872-2067(16)62522-6 shu

Selective arylation/annulation cascade reactions of 2-alkynylanilines with diaryliodonium salts

a College of Food and Drug, Luoyang Normal University, Luoyang 471934, Henan, China;
b College of Chemistry and Chemical Engineering, Henan Key Laboratory of Function-Oriented Porous Materials, Luoyang Normal University, Luoyang 471934, Henan, China

Received Date: 16 July 2016
Revised Date: 13 September 2016

Fund Project: This work was supported by the Intercollegiate Key Scientific Research Projects of Henan Province (15A150018).

An efficient Cu catalyzed selective arylation/annulation cascade reaction of 2-alkynylanilines with diaryliodonium salts was developed. This reaction was selective to N-arylation instead of C-arylation, which provides a simple synthetic method for N-aryl indoles.
- Selective arylation,
- Annulation,
- Diaryliodonium salt,
- 2-Alkynylaniline,
- N-Aryl indole,
- Cascade reaction
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