Citation: Ji Zhen LI, Xue Peng QIU, Lian Xun GAO, Meng Xian DING. Synthesis of cis-(±)-2-Hydroxymethyl-5-(Cytosine-1'-yl)- 1,3-Oxathiolane (BCH-189)[J]. Chinese Chemical Letters, ;2001, 12(6): 487-488. shu

Synthesis of cis-(±)-2-Hydroxymethyl-5-(Cytosine-1'-yl)- 1,3-Oxathiolane (BCH-189)

Polymer Chemistry Laboratory, Changchun Institute of Applied Chemistry, Chinese Academy of Sciences, Changchun 130022

Received Date: 16 October 2000

The target compound BCH-189 was synthesized with high yield via four steps from benzoyloxy acetylaldehyde and p-dithiane-2,5-diol as starting materials. The synthetic route is preferable to what literature reported.
- Anti-HIV,
- total synthesis,
- BCH-189.
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